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FOR LABORATORY RESEARCH USE ONLY — not for human or veterinary use, diagnosis, treatment, or cosmetic application. Buyers must be 21+ and legally permitted to purchase research chemicals in their jurisdiction.Intended-use statement →

Semax Wholesale

ACTH(4–7)-Pro-Gly-Pro heptapeptide — BDNF upregulation & neuroprotection research, manufacturer-direct

Product Identity

CAS Number80714-61-0
SequenceMet-Glu-His-Phe-Pro-Gly-Pro-OH
Amino Acids7 (ACTH(4-7) + Pro-Gly-Pro C-terminal)
Molecular FormulaC₃₇H₅₁N₉O₁₀S
Molecular Weight~813.9 Da
AppearanceWhite to off-white lyophilized powder
Purity≥99% by HPLC
SolubilitySoluble in sterile water or PBS
Storage2–8°C, desiccated, protect from light

Available Configurations

ConfigurationContentBest For
Standard Kit10 mg × 10 vialsNeuroprotection studies; evaluation
Bulk Kit30 mg × 10 vialsChronic cognitive models; repeat orders
CustomCustom mg × custom vialsOEM; private-label

Research Background

Semax is a synthetic heptapeptide developed at the Institute of Molecular Genetics of the Russian Academy of Sciences. It consists of the ACTH(4–7) fragment (Met-Glu-His-Phe) — the active core of adrenocorticotropic hormone that mediates neurotrophic effects without steroidogenic activity — extended with a C-terminal Pro-Gly-Pro tripeptide. Semax is the most extensively characterized nootropic peptide in the literature, with documented effects on BDNF and NGF expression, cognitive function, and neuroprotection across multiple paradigms.

Proposed Mechanisms

BDNF/NGF UpregulationEnhanced transcription of neurotrophins → synaptic plasticity
Melanocortin ReceptorMC4/MC5 receptor agonism → cAMP → CREB-mediated neurotrophin gene expression
C-terminal PGP MotifPro-Gly-Pro extension enhances metabolic stability and BBB penetration
Anti-InflammatoryReduced microglial activation; decreased IL-1β and TNF-α in CNS

Research Focus Areas

Neuroprotection

Ischemia/hypoxia models — neuronal survival enhancement

Cognitive Enhancement

Learning & memory consolidation in rodent models

BDNF/NGF Upregulation

Neurotrophin expression — synaptic plasticity support

Stroke Recovery

Post-ischemic neurological function improvement

Optic Nerve Protection

Retinal ganglion cell survival in glaucoma models

Quality Specifications

ParameterMethodCriterion
PurityHPLC at 214 nm, C18 column≥99.0% peak area
Identity (MW)ESI-MS~813.9 ± 1.0 Da
AppearanceVisual inspectionWhite to off-white powder
Peptide ContentAmino acid analysis≥80% net peptide
Met OxidationHPLC-MSMet(O) ≤ 1%

Tiered Wholesale Pricing

Kit sizeCodeList price
5 mg × 10 vialsXA5US$45
10 mg × 10 vialsXA10US$58

US$45–58 per kit (10 vials), from our published wholesale price list; tiered volume discounts apply (see the tier table) — source:wholesale price list (PDF, updated 2026-08-08).

VolumeDiscountFor
1 kitList priceEvaluation; competitive analysis
5+ kits10% offInitial portfolio expansion
20+ kits20% offMid-size distributors
50+ kits30% offRegional distributors

FAQ

What is Semax and how does it relate to ACTH?

Semax is a synthetic heptapeptide based on ACTH(4–7), the N-terminal fragment of ACTH that mediates neurotrophic effects without adrenal steroidogenesis. The C-terminal Pro-Gly-Pro extension confers metabolic stability and CNS penetration.

What is the mechanism of Semax's cognitive effects?

Semax primarily upregulates BDNF and NGF via melanocortin receptor activation. Elevated neurotrophins support synaptic plasticity, neuronal survival, and cognitive function. Additional effects include anti-inflammatory microglial modulation and improved cerebral blood flow.

How does the Pro-Gly-Pro extension work?

The C-terminal PGP tripeptide protects from carboxypeptidase degradation and enhances blood-brain barrier penetration. The Pro-Gly-Pro sequence itself has reported glyproline activity that may contribute to neuroprotection.

How does Semax differ from Selank?

Both are Russian-developed nootropics with distinct mechanisms. Semax (ACTH-derived) → melanocortin receptors → BDNF/NGF → cognition. Selank (tuftsin-derived) → GABAergic/dopaminergic → anxiolysis. Complementary: Semax for cognition, Selank for anxiety.

What purity and QC is provided for Semax?

≥99% HPLC with ESI-MS identity. Special QC: Met(O) content ≤ 1% (N-terminal methionine is oxidation-sensitive). Batch-specific COA included.

All products are manufactured for laboratory research purposes only. Semax is labeled FOR LABORATORY RESEARCH USE ONLY. Not for human or veterinary use, diagnosis, treatment, prophylaxis or any clinical, cosmetic, dietary or household application. Not a dietary supplement, pharmaceutical ingredient, cosmetic ingredient or approved drug substance. Buyers are responsible for verifying the legal status of importation and possession in their destination country.

Ready to Source Semax?

Bulk pricing, tiered discounts up to 30%, COA with every order.

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