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FOR LABORATORY RESEARCH USE ONLY — not for human or veterinary use, diagnosis, treatment, or cosmetic application. Buyers must be 21+ and legally permitted to purchase research chemicals in their jurisdiction.Intended-use statement →

GHRP-2 Wholesale

Growth Hormone Releasing Peptide-2 — potent ghrelin mimetic for GH pulse research, manufacturer-direct

Product Identity

CAS Number158861-67-7
SequenceD-Ala-D-2-Nal-Ala-Trp-D-Phe-Lys-NH₂
Amino Acids6 (D-Ala¹, D-2-Nal², D-Phe⁵)
Molecular FormulaC₄₅H₅₅N₉O₆
Molecular Weight~817.0 Da
AppearanceWhite to off-white lyophilized powder
Purity≥99% by HPLC
SolubilitySoluble in sterile or bacteriostatic water
Storage2–8°C, desiccated, protect from light

Available Configurations

ConfigurationContentBest For
Standard Kit5 mg × 10 vialsGH pulse research; evaluation
Bulk Kit10 mg × 10 vialsChronic protocols; repeat orders
CustomCustom mg × custom vialsOEM; private-label

Research Background

GHRP-2 (also known as Pralmorelin) is a synthetic hexapeptide ghrelin receptor agonist. It is one of the most potent GH secretagogues in the GHRP family, producing a rapid, robust GH pulse. Developed through structure-activity relationship studies of met-enkephalin derivatives, GHRP-2 features D-amino acid modifications (D-Ala¹, D-2-Nal², D-Phe⁵) that confer both metabolic stability and high receptor affinity.

Proposed Mechanisms

GHS-R1a AgonismPotent ghrelin receptor activation → PLC → IP₃ → Ca²⁺ mobilization → GH exocytosis
GHRH PotentiationGHS-R and GHRH-R signaling converge on somatotroph → synergistic cAMP/Ca²⁺ response
Somatostatin AntagonismGHS-R activation reduces hypothalamic somatostatin release → permissive GH secretion

Research Focus Areas

GH Pulse Induction

Rapid, potent GH release via GHS-R1a activation on pituitary

Pulsatile GH Research

Sharp GH spikes — compatible with post-exercise window protocols

Appetite Signaling

Ghrelin pathway activation — feeding behavior studies

IGF-1 Axis

GH-mediated hepatic IGF-1 production cascade

Quality Specifications

ParameterMethodCriterion
PurityHPLC at 214 nm, C18 column≥99.0% peak area
Identity (MW)ESI-MS~817.0 ± 1.0 Da
AppearanceVisual inspectionWhite to off-white powder
Chiral PurityChiral HPLCD-amino acids verified
Residual MoistureKarl Fischer≤3%

Tiered Wholesale Pricing

Kit sizeCodeList price
5 mg × 10 vialsG25US$42

US$42–42 per kit (10 vials), from our published wholesale price list; tiered volume discounts apply (see the tier table) — source:wholesale price list (PDF, updated 2026-08-08).

VolumeDiscountFor
1 kitList priceEvaluation; competitive analysis
5+ kits10% offInitial portfolio expansion
20+ kits20% offMid-size distributors
50+ kits30% offRegional distributors

FAQ

How potent is GHRP-2 vs other GH secretagogues?

GHRP-2 is among the most potent GHS-R1a agonists, producing GH elevations exceeding GHRP-6 and Ipamorelin at equivalent doses. However, this potency comes with broader receptor profile including stronger appetite stimulation.

What distinguishes GHRP-2 from Ipamorelin?

GHRP-2: more potent GH release, stronger hunger signaling, potential cortisol elevation. Ipamorelin: cleaner GH pulse, minimal hunger, minimal cortisol. Choice depends on whether maximum amplitude or receptor selectivity is the priority.

What is the origin of GHRP-2?

GHRP-2 (Pralmorelin) was developed by Kaken Pharmaceutical in Japan through systematic modification of met-enkephalin derivatives. D-amino acid substitutions provide enzymatic resistance while maintaining high GHS-R1a binding affinity.

How should GHRP-2 be stored?

Lyophilized: 2–8°C, desiccated, 24-month stability. After reconstitution, aliquot and store at -20°C. Avoid freeze-thaw cycles. D-amino acid modifications provide good solution stability.

Can GHRP-2 be combined with CJC-1295?

Yes — common research combination. CJC-1295 provides sustained GHRH signal; GHRP-2 provides potent ghrelin receptor pulse. CJC-1295 (no DAC) + GHRP-2 is particularly suited for pulsatile GH protocol research.

All products are manufactured for laboratory research purposes only. GHRP-2 is labeled FOR LABORATORY RESEARCH USE ONLY. Not for human or veterinary use, diagnosis, treatment, prophylaxis or any clinical, cosmetic, dietary or household application. Not a dietary supplement, pharmaceutical ingredient, cosmetic ingredient or approved drug substance. Buyers are responsible for verifying the legal status of importation and possession in their destination country.

Ready to Source GHRP-2?

Bulk pricing, tiered discounts up to 30%, COA with every order.

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